Halotestin 10 mg

ACTIVE INGREDIENT

Each tablet contains:Fluoxymesterone 10 mg

DESCRIPTION

Fluoxymesterone, marketed as Halotestin, is a synthetic androgenic anabolic steroid. It is primarily used in the treatment of conditions related to low testosterone levels in males, delayed puberty, and certain types of breast cancer in women. Known for its potent anabolic properties, Fluoxymesterone is effective in promoting muscle growth and enhancing physical performance, making it popular among athletes and bodybuilders.

PHARMACOLOGICAL PROPERTIES

Mechanism of Action:
Fluoxymesterone binds to androgen receptors, stimulating protein synthesis and promoting muscle growth. It also has antitumor effects by blocking the growth of certain breast cancer cells.Pharmacokinetics:

• Absorption: Oral absorption is approximately 80%.
• Distribution: Highly protein-bound (99%), primarily to sex hormone-binding globulin.
• Metabolism: Metabolized in the liver.
• Half-life: Approximately 9.2 hours.
• Excretion: Eliminated mainly through urine.

INDICATIONS

Fluoxymesterone is indicated for:

• Hypogonadism: Replacement therapy for males with low testosterone levels.
• Delayed puberty: Treatment in boys diagnosed with delayed puberty.
• Breast cancer: Palliative treatment for hormone-responsive recurrent breast cancer in postmenopausal women.

DOSAGE AND ADMINISTRATION

Dosage:

• Usual Adult Dose for Hypogonadism: 10 to 40 mg per day, divided into multiple doses.
• Usual Pediatric Dose for Delayed Puberty: Individualized based on weight and clinical response.

Administration:
Take orally with or without food, as directed by a healthcare provider.

CONTRAINDICATIONS

• Hypersensitivity to Fluoxymesterone or any formulation component.
• Pregnancy (Pregnancy Category X).
• Active breast or prostate cancer in males.
• Severe liver dysfunction.

WARNINGS AND PRECAUTIONS

1. Hepatic Effects: Potential for severe liver toxicity; regular monitoring of liver function is recommended.
2. Cardiovascular Risks: May increase cholesterol levels and risk of cardiovascular events; monitor lipid profiles regularly.
3. Androgenic Effects: Possible side effects include acne, hair loss, and virilization in women; caution is advised for female patients.
4. Fluid Retention: Can cause edema; monitor for signs such as rapid weight gain or shortness of breath.

ADVERSE REACTIONS

Common Adverse Reactions:

• Acne
• Mood changes
• Insomnia
• Swelling

Serious Adverse Reactions:

• Liver damage: Symptoms may include jaundice and abdominal pain.
• Cardiovascular issues: Increased risk of heart attack or stroke.
• Hormonal imbalances: Gynecomastia in men and virilization symptoms in women.

INTERACTIONS

1. Anticoagulants: May enhance anticoagulant effects, increasing bleeding risk; monitor coagulation parameters closely.
2. Corticosteroids: Concurrent use may increase fluid retention risk.

USE IN SPECIFIC POPULATIONS

• Pregnancy and Lactation: Contraindicated due to potential teratogenic effects.
• Pediatric Use: Use with caution due to risks of growth interference and hormonal imbalance.
• Geriatric Use: Caution advised due to increased risk of adverse effects related to cardiovascular health and liver function.

OVERDOSAGE

There is no specific antidote for Fluoxymesterone overdose. Supportive care and symptomatic treatment are recommended while monitoring liver and cardiovascular function closely.

STORAGE

Store below 25°C (77°F). Protect from light. Keep out of reach of children.

PACKAGING

Fluoxymesterone 10 mg is supplied as oral tablets in various packaging configurations.

MANUFACTURER

Oxydine Metabolics Switzerland

Oxydine.org
Hi@Oxydine.org